Enzyme Inhibitors
Enzyme inhibitors are molecules that bind to enzymes and decrease their activity. Since blocking an enzyme’s activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors.The binding of an inhibitor can stop a substrate from entering the enzyme’s active site and/or hinder the enzyme from catalysing its reaction. Inhibitor binding is either reversible or irreversible. Irreversible inhibitors usually react with the enzyme and change it chemically.
Sub-categories for Enzyme Inhibitors Category
Showing 121–132 of 310 results
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VD-OEIA-0033
GSK-3 Inhibitor IX
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Appearance:
Dark red solid
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CAS Number:
710323-61-8
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Cat.number:
VD-OEIA-0033
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Formula:
C17H12BrN3O2
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VD-OEIA-0016
GSK-3 Inhibitor X
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Appearance:
Dark purple solid
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CAS Number:
740841-15-0
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Cat.number:
VD-OEIA-0016
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Formula:
C18H12BrN3O3
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VD-OEIA-00177
GSK-3 Inhibitor XV
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Appearance:
Purple solid
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CAS Number:
N/A
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Cat.number:
VD-OEIA-00177
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Formula:
C25H14BrN3O6Ru
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VD-OEIA-0018
GSK-3β Inhibitor I
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Appearance:
White Solid
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CAS Number:
327036-89-5
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Cat.number:
VD-OEIA-0018
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Formula:
C10H10N2SO2
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VD-OEIA-0218
GSK-3β Inhibitor II (CAS 478482-75-6)
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Appearance:
Yellow solid.
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CAS Number:
478482-75-6
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Cat.number:
VD-OEIA-0218
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Formula:
C14H10IN3OS
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VD-OEIA-0019
GSK-3β Inhibitor VI
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Appearance:
Orange solid
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CAS Number:
62673-69-2
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Cat.number:
VD-OEIA-0019
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Formula:
C6H3Br2ClOS
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VD-OEIA-0020
GSK-3β Inhibitor VII
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Appearance:
White Solid
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CAS Number:
99-73-0
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Cat.number:
VD-OEIA-0020
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Formula:
C8H6Br2O
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VD-OEIA-0032
GSK-3β Inhibitor VIII
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Appearance:
Off-white to tan powder.
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CAS Number:
487021-52-3
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Cat.number:
VD-OEIA-0032
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Formula:
C12H12N4O4S
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VD-OEIA-00222
GSK-3β Inhibitor XI
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Appearance:
Orange red solid
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CAS Number:
626604-39-5
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Cat.number:
VD-OEIA-00222
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Formula:
C18H15N5O3
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VD-PI-0094
GW 9662 (CAS 22978-25-2)
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Appearance:
Off-white solid
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CAS Number:
22978-25-2
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Cat.number:
VD-PI-0094
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Formula:
C13H19N2O3Cl
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VD-OEIA-1094
GW4869
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Appearance:
Pale yellow solid.
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CAS Number:
6823-69-4
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Cat.number:
VD-OEIA-1094
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Formula:
C30H28N6O2 . 2HCl
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VD-OEIA-0035
H-ILE-AMC TFA
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Appearance:
White to off-white powder
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CAS Number:
191723-68-9
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Cat.number:
VD-OEIA-0035
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Formula:
C18H21F3N2O5
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