CARTProduct Variations
| Product # | Price | Quantity | |
|---|---|---|---|
| VD-OEIA-1072-0005-5mg | $125 | ||
| VD-OEIA-1072-0025-25mg | $450 |
GDC-0941 bismesylate
$125.00 – $450.00
Product Specification
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Appearance:
N/A
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CAS Number:
957054-30-7
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Cat.number:
VD-OEIA-1072
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Formula:
C23H27N7O3S2.2CH3SO3H
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MW:
705.83
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Purity:
>=98%
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Solubility:
DMSO and water.
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Storage:
-20°C.Protect from light.
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Synonyms:
4-(2-(1H-indazol-4-yl)-6-((4-(methylsulfonyl)piperazin-1-yl)methyl) thieno[3,2-d]pyrimidin-4-yl)morpholine dimethanesulfonate
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Size:
25mg, 5mg
Description
Potent, selective, orally bioavailable inhibitor of class I PI3 kinase (PI3K) under clinical trials, with IC50 values (nM) of 3, 33, 3, 75, 1230 and 580 for p110 α, β, δ and γ isoforms, DNA-PK and mTOR.
1.AJ Folkes et al. J. Med. Chem. (2008), 51(18), 5522-32.
2.FI Raynaud et al. Mol. Cancer Ther. (2009), 8(7), 1725-38.
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