CARTProduct Variations
| Product # | Price | Quantity | |
|---|---|---|---|
| VD-OEIA-0019-0005-5mg | $70 | ||
| VD-OEIA-0019-0050-50mg | $600 |
GSK-3β Inhibitor VI
$70.00 – $600.00
Product Specification
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Appearance:
Orange solid
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CAS Number:
62673-69-2
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Cat.number:
VD-OEIA-0019
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Formula:
C6H3Br2ClOS
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MW:
318.41
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Purity:
≥90%
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Solubility:
DMSO or EtOH
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Storage:
-20°C
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Synonyms:
2-chloro-1-(4,5-dibromothiophen-2-yl)ethanone
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Size:
50mg, 5mg
Description
A thienyl α-chloromethyl ketone compound that acts as a cell-permeable, irreversible, and non-ATP competitive inhibitor of GSK-3β (IC50 = 1 µM). This reactive alkylating agent is selective towards GSK-3β and does not affect PKA activity even at concentrations as high as 100 µM.
1.Conde, S., et al. 2003. J. Med. Chem. 46, 4631.
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