CARTProduct Variations
| Product # | Price | Quantity | |
|---|---|---|---|
| VD-OEIA-1012-0005-5mg | $120 | ||
| VD-OEIA-1012-0025-25mg | $500 |
Rho Kinase Inhibitor V
$120.00 – $500.00
Product Specification
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Appearance:
Light beige solid.
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CAS Number:
1072906-02-5
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Cat.number:
VD-OEIA-1012
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Formula:
C18H15N3O3
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MW:
321.3
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Purity:
>=97% by (HPLC)
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Solubility:
DMSO or EtOH.
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Storage:
+2°C to +8°C. Protect from light.
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Synonyms:
N/A
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Size:
25mg, 5mg
Description
A cell-permeable pyrazolyl carboxamide compound that acts as a potent, ATP-binding pocket-targeting inhibitor of ROCK-II and effectively inhibits the myosin light chain 2 phosphorylation on Thr18/Ser19 in A7r5 cells. It affects the activities of PKA, MRCK, Akt1 and CYP-450 enzymes only at much higher concentrations.
1.Feng, Y., et al. 2008. J. Med. Chem. 51, 6642.
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