CARTProduct Variations
| Product # | Price | Quantity | |
|---|---|---|---|
| VD-OEIA-1086-0010-10mg | $170 | ||
| VD-OEIA-1086-0050-50mg | $600 |
SDZ NKT 343
$170.00 – $600.00
Product Specification
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Appearance:
Yellow solid.
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CAS Number:
180046-99-5
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Cat.number:
VD-OEIA-1086
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Formula:
C33H33N5O5
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MW:
579.65
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Purity:
>=98%
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Solubility:
100 mM in DMSO and to 100 mM in Ethanol.
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Storage:
+2°C to +4°C. Protect from light.
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Synonyms:
N/A
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Size:
10mg, 50mg
Description
Highly selective human tachykinin NK1 receptor antagonist (IC50 values are 0.62 and 451 nM for human and rat receptors respectively) that displays > 130-fold selectivity over human NK2 and NK3 receptors. Potently antagonizes SP-induced Ca2+ efflux in vitro and inhibits mechanical hyperalgesia in vivo.
1.Walpole et al (1998), J.Med.Chem. 41 3159.
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