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MRS 5698 (CAS 1377273-00-1)




Product specification

Formula: C28H23ClF2N6O3
MW: 564.97
Purity: >=96%
Appearance: White solid
Solubility: 10 mM in DMSO.
Storage: -20°C.
CAS Number: 1377273-00-1
Synonyms: MRS5698
Cat.number: VD-TMR-0013

Product Description

MRS 5698 (CAS 1377273-00-1) is a high affinity and selective A3 adenosine receptor agonist (Ki ~ 3 nM); displays >1000-fold selectivity over A1 and A2A adenosine receptors. Reverses mechanoallodynia in several neuropathic pain models in vivo. Orally bioavailable.



Product References
1. Tosh et al (2012) J.Med.Chem. 55 4847.
2. Little et al (2015) Brain 138 28.