CARTProduct Variations
| Product # | Price | Quantity | |
|---|---|---|---|
| VD-AM-0100-0010-10mg | $70 | ||
| VD-AM-0100-0050-50mg | $325 |
PD 166793 (CAS 199850-67-4)
$70.00 – $325.00
Product Specification
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Appearance:
Off-white solid
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CAS Number:
199850-67-4
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Cat.number:
VD-AM-0100
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Formula:
C17H18BrNO4S
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MW:
412.3
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Purity:
≥98% by TLC
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Solubility:
100 mM in DMSO and to 100 mM in Ethanol
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Storage:
+2°C to +8°C. Protect from light.
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Synonyms:
Not available.
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Size:
10mg, 50mg
Description
PD 166793 (CAS 199850-67-4) is a cell-permeable biphenylsulfonylvaline compound that acts as a potent inhibitor against MMP-2, -3, and -13 (IC50 = 47, 12, and 8 nM, respectively) and a weaker inhibitor against AMP deaminase (20% inhibition at 0.1 µM), MMP-1, -7, -9, and -14 (IC50 = 6.1, 7.2, 7.9, and 0.24 µM, respectively). Shown to offer therapeutic benefits in vivo in various animal models of heart failure and diabetes.
1.O’Brien et al (2000). J.Med.Chem. 43 156.
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